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1039825-68-7 | MCH-1 antagonist 1

MCH-1 antagonist 1 NLT 98%

SKU : MC503671

CAS Number : 1039825-68-7

Molecular Formula : C25H26N4O2 | Molecular Weight : 414.50

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Purity NLT 98%
Storage at 20ºC 2 years

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Chemical Name MCH-1 antagonist 1
CAS Number 1039825-68-7
MDL Number MFCD18633193
Molecular Formula C25H26N4O2
Molecular Weight 414.50
Introduction of 1039825-68-7 :

MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist with a Ki of 2.6 nM. MCH-1 antagonist 1 also inhibits CYP3A4 with an IC50 of 10 μM. IC50 & Target: Ki: 2.6 nM (MCH-1)[1]
IC50: 10 μM (CYP3A4)[1] In Vitro: MCH-1 antagonist 1 (Compound 1) also inhibits cytochrome P450 3A4 (CYP3A4) with an IC50 of 10 μM[1]. In Vivo: MCH-1 antagonist 1 is administered to male C57BL/6J DIO mice to assess their pharmacokinetic profile. Effect of MCH-1 antagonist 1 (dosed at 30 mg/kg, po) is measured on the body weight of DIO mice with the AUC0-6 h of 14760 h*ng/mL[1].

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