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109826-27-9 | Zaldaride maleate

Zaldaride maleate NLT 98%

SKU : MC506116

CAS Number : 109826-27-9

Molecular Formula : C30H32N4O6 | Molecular Weight : 544.60

Synonyms : CGS-9343B;KW 5617

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Purity NLT 98%
Storage at 20ºC 2 years

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Chemical Name Zaldaride maleate
CAS Number 109826-27-9
MDL Number MFCD04113002
Molecular Formula C30H32N4O6
Molecular Weight 544.60
Synonyms CGS-9343B;KW 5617
Introduction of 109826-27-9 :

Zaldaride maleate (CGS-9343B) is a potent, orally active and selective inhibitor of calmodulin. Zaldaride maleate (CGS-9343B) inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity, with an IC50 of 3.3 nM[1][2]. Zaldaride maleate (CGS-9343B) prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+ and K+ currents in PC12 cells and inhibits nAChR[3]. IC50 & Target: IC50: 3.3 nM (calmodulin)[1][2]. In Vivo: Zaldaride maleate (KW 5617, P.O., 3 mg/kg) ameliorates the diarrhea in the 16, 16-dimethyl prostaglandin E2 model[4].

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