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1000690-85-6 | Tilapertin

Tilapertin NLT 98%

Product Number : MC500236

CAS Number : 1000690-85-6

Molecular Formula : C20H21F3N2O2 | Molecular Weight : 378.39

Synonyms : AMG747

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Purity NLT 98%
Storage at 20ºC 2 years
MolCore specializes in manufacturing high-purity CAS No.1000690-85-6, Tilapertin with the molecular formula C20H21F3N2O2 and molecular weight 378.39 delivering critical API intermediates for global pharmaceutical and research industries, certified under ISO quality systems.

* The above information is for reference only.

Chemical Name Tilapertin
CAS Number 1000690-85-6
Molecular Formula C20H21F3N2O2
Molecular Weight 378.39
Synonyms AMG747
Introduction of 1000690-85-6 :

Tilapertin is an oral inhibitor of glycine transporter type-1 (GlyT1). IC50 & Target: GlyT1[1] In Vivo: Tilapertin is a nanomolar potent, orally bioavailable and selective GlyT1 inhibitor. Oral administration of Tilapertin dose-dependently increases cerebrospinal fluid (CSF) glycine concentration in rats[1].