SKU : MC501614
CAS Number : 1011531-27-3
Molecular Formula : C24H19F3N2O4S | Molecular Weight : 488.48
Quote RequestPurity | NLT 98% |
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Storage | at 20ºC 2 years |
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Chemical Name | AM-4668 |
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CAS Number | 1011531-27-3 |
Molecular Formula | C24H19F3N2O4S |
Molecular Weight | 488.48 |
AM-4668 is a GPR40 agonist for type 2 diabetes. EC50s of 3.6 nM and 36 nM for GPR40 in A9 cells (GPR40 IP3 assay) and CHO cells (GPR40 aequorin assay), respectively[1]. IC50 & Target: EC50: 3.6 nM (GPR40, in A9 cells), 36 nM (GPR40, in CHO cells)[1]
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