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1021868-83-6 | ARL67156 trisodium salt

ARL67156 trisodium salt NLT 98%

SKU : MC502544

CAS Number : 1021868-83-6

Molecular Formula : C15H21Br2N5Na3O12P3 | Molecular Weight : 785.05

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Purity NLT 98%
Storage at 20ºC 2 years

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Chemical Name ARL67156 trisodium salt
CAS Number 1021868-83-6
Molecular Formula C15H21Br2N5Na3O12P3
Molecular Weight 785.05
Introduction of 1021868-83-6 :

ARL67156 trisodium salt is an inhibitor of ecto-ATPase. ARL 67156 is a weak competitive inhibitor of NTPDase1 (CD39), NTPDase3 and NPP1, with Kis of 11, 18 and 12 μM, respectively[1]. IC50 & Target: Ki: 11 μM (NTPDase1), 18 μM (NTPDase3), 12 μM (NPP1)[1] In Vitro: ARL67156 trisodium salt is also an effective inhibitor of UTP breakdown by superior cervical ganglion cells and to potentiate contractions elicited by this nucleotide in isolated tail artery of rat. ARL67156 is not an effective inhibitor of NTPDase2, NTPDase8, NPP3 and ecto-5′-nucleotidase (CD73), although it also reduces the activity of these enzymes[1].

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