SKU : MC507221
CAS Number : 112748-19-3
Molecular Formula : C77H119N21O26S3 | Molecular Weight : 1851.09
Quote RequestPurity | NLT 98% |
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Storage | at 20ºC 2 years |
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Chemical Name | Scyliorhinin II |
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CAS Number | 112748-19-3 |
MDL Number | MFCD00080018 |
Molecular Formula | C77H119N21O26S3 |
Molecular Weight | 1851.09 |
Scyliorhinin II is a selective neurokinin-3 receptor agonist, with a Ki of 2.5 nM for neurokinin-3 receptor in rat cerebral cortex. IC50 & Target: Ki: 2.5 nM (Neurokinin-3 receptor)[1] In Vitro: Scyliorhinin II is a neurokinin-3 selective tachykinin receptor, with a Ki of 2.5 nM for neurokinin-3 (NK-3) receptor in rat cerebral cortex. Scyliorhinin II has little effect on NK-1 and NK-2 receptors, with Ki (NK-1 receptor)/Ki (NK-3 receptor) and Ki (NK-2 receptor)/Ki (NK-3 receptor) of 176 and 200[1]. In Vivo: Scyliorhinin II produces potent, dose-related reciprocal hindlimb scratching about equipotently with an ED50 of 0.08 nmol via intracerebroventricularly (i.c.v.) administration in mice[2].
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