SKU : MC531307
CAS Number : 171714-84-4
Molecular Formula : C22H22N2O6 | Molecular Weight : 410.42
Synonyms : Lu-135252
Quote RequestPurity | NLT 98% |
---|---|
Storage | at 20ºC 2 years |
* The above information is for reference only.
* If the product has intellectual property rights, a license granted is must or contact us.
Chemical Name | Darusentan |
---|---|
CAS Number | 171714-84-4 |
MDL Number | MFCD00949063 |
Molecular Formula | C22H22N2O6 |
Molecular Weight | 410.42 |
Synonyms | Lu-135252 |
Darusentan is a selective endothelin A (ETA) receptor antagonist. Darusentan competes for radiolabeled endothelin binding in rat aortic vascular smooth muscle cells (RAVSMs) membranes with single-site kinetics, exhibiting a Ki=13 nM[1].
© Copyright 2015-2024 Hangzhou MolCore BioPharmatech Co.,Ltd. All rights reserved.