SKU : MC537769
CAS Number : 201038-74-6
Molecular Formula : C18H28N2O3S | Molecular Weight : 352.49
Quote RequestPurity | NLT 98% |
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Storage | at 20ºC 2 years |
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Chemical Name | SB-269970 |
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CAS Number | 201038-74-6 |
MDL Number | MFCD08056273 |
Molecular Formula | C18H28N2O3S |
Molecular Weight | 352.49 |
SB269970 is a 5-HT7 receptor antagonist with pKi of 8.3, exhibits >50-fold selectivity against other receptors. IC50 & Target: pKi: 8.3 (5-HT7 receptor)[1] In Vivo: SB-269970 (3-30 mg/kg; i.p.; once) significantly blocks amphetamine and ketamine-induced hyperactivity[2].
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