Product Number : MC544400
CAS Number : 251945-92-3
Molecular Formula : C18H20N4O | Molecular Weight : 308.38
Synonyms : SLV 320
Quote RequestPurity | NLT 98% |
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Storage | at 20ºC 2 years |
MolCore specializes in manufacturing high-purity CAS No.251945-92-3, Derenofylline with the molecular formula C18H20N4O and molecular weight 308.38 delivering critical API intermediates for global pharmaceutical and research industries, certified under ISO quality systems. |
* The above information is for reference only.
Chemical Name | Derenofylline |
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CAS Number | 251945-92-3 |
MDL Number | MFCD12756289 |
Molecular Formula | C18H20N4O |
Molecular Weight | 308.38 |
Synonyms | SLV 320 |
Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1]. IC50 & Target: Ki: 1 nM (adenosine A1 receptor)[1].
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