Product Number : MC545315
CAS Number : 264622-58-4
Molecular Formula : C26H26N6O4 | Molecular Weight : 486.52
Quote RequestPurity | NLT 98% |
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Storage | at 20ºC 2 years |
MolCore specializes in manufacturing high-purity CAS No.264622-58-4, MRS 1754 with the molecular formula C26H26N6O4 and molecular weight 486.52 delivering critical API intermediates for global pharmaceutical and research industries, certified under ISO quality systems. |
* The above information is for reference only.
Chemical Name | MRS 1754 |
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CAS Number | 264622-58-4 |
MDL Number | MFCD09971130 |
Molecular Formula | C26H26N6O4 |
Molecular Weight | 486.52 |
MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats[1]. IC50 & Target: A2B Adenosine Receptor[1] In Vitro: The most potent displacer of [3H]MRS 1754 binding is MRS 1754. The Ki value for displacement of [3H]MRS 1754 binding to human A2B receptors expressed in HEK-293 cell membranes is 1.45±0.21 nM[1].
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